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首次探索喹硫平(Quetiapine,QUE)原料及片剂氧化降解产生的新分子 ...
喹硫平(QUE)是 FDA 批准的抗躁狂和抗精神分裂活性药物成分,其片剂稳定性需关注,杂质或降解产物允许量有规定。研究人员探索其降解途径,对氧化降解产物进行研究。结果发现新降解产物有抗菌活性,也有不良影响。该研究为新抗菌剂提供潜在支架。
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