Pregabalin binds with high affinity to the alpha2 ... Peak plasma concentration: 1.5 hours (capsules). Oral bioavailability: ≥90%. Steady state: achieved within 24–48 hours.

Conversion from Lyrica capsules, oral soln: see full labeling. For all: renal impairment (CrCl 30–60mL/min): reduce dose (see full labeling); (CrCl <30mL/min or hemodialysis): dose with Lyrica.